1. Junshan Tian, Jiankang Zhong, Yunsheng Li, and Dawei Ma*, Organocatalytic and Scalable Synthesis of the Anti-Influenza Drugs Zanamivir, Laninamivir, and CS-8958. Angewandte Chemie, International Edition, 2014, 53, 13885-13888.
  2.  Mingxing Teng, Weiwei Zi, and Dawei Ma*, Total Synthesis of the Monoterpenoid Indole Alkaloid (±)-Aspidophylline A. Angewandte Chemie, International Edition, 2014, 53, 1814-11817.
  3. Chengang Zhou and Dawei Ma*, A copper-catalyzed coupling reaction of vinyl halides and carbazates: application in the assembly of polysubstituted pyrroles, Chemical Communications, 2014, 50, 3085-3088.
  4. Huan Liu, Guangde Jiang, Xixian Pan, Xiaolong Wan, Yisheng Lai, Dawei Ma*, and Weiqing Xie, Highly Asymmetric Bromocyclization of Tryptophol: Unexpected Accelerating Effect of DABCO-Derived Bromine Complex, Organic Letters 2014, 16, 1908-1911.
  5. Wu, Mingyao; Ma, Dawei *Total Syntheses of (±)-Spiroquinazoline, (-)-Alantryphenone, (+)-Lapatin A, and (-)-Quinadoline B. Angewandte Chemie, International Edition 2013, 52, 9759-9762.
  6. Xie Weiqing; Jiang Guangde; Liu Huan; Hu Jiadong; Pan Xixian; Zhang Hui; Wan Xiaolong; Lai Yisheng; Ma Dawei* Highly Enantioselective Bromocyclization of Tryptamines and Its Application in the Synthesis of (-)-Chimonanthine. Angewandte Chemie, International edition 2013, 52, 12924-12927.
  7. Wei, Yi; Zhao, Duo; Ma, Dawei *Total Synthesis of the Indole Alkaloid (±)- and (+)-Methyl N-Decarbomethoxychanofruticosinate. Angewandte Chemie, International Edition, 2013, 52, 12988-12991.
  8. Fan, Mengyang; Ma, Dawei *Palladium-Catalyzed Direct Functionalization of 2-Aminobutanoic Acid Derivatives: Application of a Convenient and Versatile Auxiliary. Angewandte Chemie, International Edition 2013, 52(46), 12152-12155
  9. Xie, Weiqing; Zuo, Zhiwei; Zi, Weiwei; Ma, Dawei*  Intramolecular oxidative coupling: applications in synthesis of complex indole akaloid scaffolds Youji Huaxue 2013, 33(5), 869-876.
  10. Jiang, Yongwen; Xu, Lanting; Zhou, Chenggang; Ma, Dawei* Cu-catalyzed Ullmann-type C-heteroatom bond formation: the key role of dinucleating ancillary ligands RSC Catalysis Series 2013, 11(C-H and C-X Bond Functionalization), 1-45.
  11. Chen, Yu; Lu, Yuwei; Zou, Qing; Chen, Huansheng; Ma, Dawei*  A Scalable Process to the Key Intermediate of Cilazapril, (S)-1-Benzyloxycarbonylhexahydropyridazine-3-carboxylic Acid, Through a Novel Cascade Course Organic Process Research & Development 2013, 17(9), 1209-1213.
  12. Xie, Weiqing; Wang, Hexiang; Fan, Feng; Tian, Junshan; Zuo, Zhiwei; Zi, Weiwei; Gao, Kun; Ma, Dawei* Diastereoselective construction of continuous all-carbon quaternary centers via intramolecular oxidative coupling reaction Tetrahedron Letters 2013, 54(33), 4392-4396.
  13. Kishor, Chandan; Arya, Tarun; Reddi, Ravikumar; Chen, Xiaochun; Saddanapu, Venkateshwarlu; Marapaka, Anil Kumar; Gumpena, Rajesh; Ma, Dawei*; Liu, Jun O.; Addlagatta, Anthony Identification, Biochemical and Structural Evaluation of Species-Specific Inhibitors against Type I Methionine Aminopeptidases Journal of Medicinal Chemistry 2013, 56(13), 5295-5305.
  14. Xie, Siwei; Qin, Peng; Li, Meng; Zhang, Xiaojing; Jiang, Yongwen; Ma, Dawei* Synthesis of 2-alkyl-2-arylcyanoacetates via CuI/sodium picolinate-catalyzed direct arylation of a-substituted cyanoacetates Tetrahedron Letters 2013, 54(29), 3889-3891.
  15. Yin, Hongfei; Chen, Bing; Zhang, Xiaojing; Yang, Xinye; Zhang, Yihua; Jiang, Yongwen; Ma, Dawei* Assembly of N,N-disubstituted-N'-arylureas via a copper-catalyzed one-pot three-component reaction of aryl bromides, potassium cyanate, and secondary amines Tetrahedron 2013, 69(26), 5326-5330.
  16. Zhang, Pengtao; Yang, Xinye; Zhang, Feiran; Gabelli, Sandra B.; Wang, Renxiao; Zhang, Yihua; Bhat, Shridhar; Chen, Xiaochun; Furlani, Manuel; Amzel, L. Mario; et al  Pyridinylpyrimidines selectively inhibit human methionine aminopeptidase-1 Bioorganic & Medicinal Chemistry 2013, 21(9), 2600-2617.
  17. Xu, Lanting; Peng, Yinsheng; Pan, Qiangbiao; Jiang, Yongwen; Ma, Dawei *Assembly of Substituted 3-Aminoindazoles from 2-Bromobenzonitrile via a CuBr-Catalyzed Coupling/Condensation Cascade Process Journal of Organic Chemistry 2013, 78(7), 3400-3404.
  18. Zhang, Ye; Xing, Hui; Xie, Weiqing; Wan, Xiaolong; Lai, Yisheng; Ma, Dawei* Asymmetric, Regioselective Bromohydroxylation of 2-Aryl-2-propen-1-ols Catalyzed by Quinine-Derived Catalysts Advanced Synthesis & Catalysis 2013, 355, 68-72. 
  19. Zhang, Feiran; Bhat, Shridhar; Gabelli, Sandra B.; Chen, Xiaochun; Miller, Michelle S.; Nacev, Benjamin A.; Cheng, Yim Ling; Meyers, David J.; Tenney, Karen; Shim, Joong Sup; Crews, Phillip; Amzel, L. Mario; Ma, Dawei*; Liu, Jun O. Pyridinylquinazolines Selectively Inhibit Human Methionine Aminopeptidase-​1 in Cells Journal of Medicinal Chemistry 2013, 56, 3996-4016.
  20. Songchuan Tian, Weiwei Zi, Dawei Ma* ‘Potentially Biomimetic Total Synthesis and Relative Stereochemical Assignment of (±)-Gracilamine’ Angewandte Chemie, International Edition 2012, 51(40), 10141-10144
  21. Fan, Feng; Xie, Weiqing; Ma, Dawei* Cascade annulation of malonic diamides: a concise synthesis of polycyclic pyrroloindolines, Chemical Communications (Cambridge, United Kingdom) 2012, 48, 7571-7573.
  22. Fan, Feng; Xie, Weiqing; Ma, Dawei* Construction of Polycyclic Spiro-indolines via an Intramolecular Oxidative Coupling/Cyclization Cascade Reaction Process, Organic Letters 2012, 14, 1405-1407.
  23. Huo, Lele; Ma, Anqi; Zhang, Yihua; Ma, Dawei* Assembly of 4-Substituted 3-Nitro-1,2,3,4-tetrahydropyridines via Organocatalytic Michael Addition, Advanced Synthesis & Catalysis 2012, 354, 991-994.
  24. Li, Jiaojiao; Zhang, Yihua; Jiang, Yongwen; Ma, Dawei* CuI/N,N-dimethylglycine-catalyzed synthesis of N-aryloxazolidinones from aryl bromides, Tetrahedron Letters 2012, 53, 3981-3983.
  25. Li, Jiaojiao; Zhang, Yihua; Jiang, Yongwen; Ma, Dawei* CuI-catalyzed one-pot synthesis of benzothiazolones from 2-iodoanilines-derived carbamates and sodium sulfide, Tetrahedron Letters 2012, 53, 2511-2513.
  26. Liu, Qing; Li, Na; Yuan, Yunyun; Lu, Huili; Wu, Xiaoyan; Zhou, Caihong; He, Min; Su, Haoran; Zhang, Meng; Wang, Jia; Wang, Bao; Wang, You; Ma, Dawei*; Ye, Yang; Weiss, Hans-Christoph; Gesing Ernst, R. F.; Liao, Jiayu; Wang, Ming-Wei Cyclobutane derivatives as novel nonpeptidic small molecule agonists of glucagon-like peptide-1 receptor, J Med Chem 2012, 55, 250-267.
  27. Wang, Leilei; Zhang, Xiaojing; Ma, Dawei* Organocatalytic Michael addition of aldehydes to trisubstituted nitroolefins, Tetrahedron 2012, 68, 7675-7679.
  28. Xing, Hui; Zhang, Ye; Lai, Yisheng; Jiang, Yongwen; Ma, Dawei* Synthesis of Symmetrical and Unsymmetrical N,N'-Diaryl Guanidines via Copper/N-Methylglycine-Catalyzed Arylation of Guanidine Nitrate, Journal of Organic Chemistry 2012, 77, 5449-5453.
  29. Xiong, Xiaodong; Jiang, Yongwen; Ma, Dawei* Assembly of N,N-Disubstituted Hydrazines and 1-Aryl-1H-indazoles via Copper-Catalyzed Coupling Reactions, Organic Letters 2012, 14, 2552-2555.
  30. Xu, Lanting; Jiang, Yongwen; Ma, Dawei* Synthesis of 3-Substituted and 2,3-Disubstituted Quinazolinones via Cu-Catalyzed Aryl Amidation, Organic Letters 2012, 14, 1150-1153.
  31. Yang, Xinye; Xing, Hui; Zhang, Ye; Lai, Yisheng; Zhang, Yihua; Jiang, Yongwen; Ma, Dawei* CuI/8-Hydroxyquinaldine Promoted N-Arylation of Indole and Azoles, Chinese Journal of Chemistry 2012, 30, 875-880.
  32. Zhang, Yu; Yang, Xinye; Yao, Qizheng; Ma, Dawei* CuI/DMPAO-Catalyzed N-Arylation of Acyclic Secondary Amines, Organic Letters 2012, 14, 3056-3059.
  33. Zi, Weiwei; Xie, Weiqing; Ma, Dawei* Total Synthesis of Akuammiline Alkaloid (-)-Vincorine via Intramolecular Oxidative Coupling, Journal of the American Chemical Society 2012, 134, 9126-9129.
  34. Chen, Gang; Xia, Hongguang; Cai, Yu; Ma, Dawei*; Yuan, Junying; Yuan, Chengye Diphenylbutylpiperidine-based cell autophagy inducers: Design, synthesis and SAR studies, MedChemComm 2011, 2, 315-320.
  35. Chen, Gang; Xia, Hongguang; Cai, Yu; Ma, Dawei*; Yuan, Junying; Yuan, Chengye Synthesis and SAR study of diphenylbutylpiperidines as cell autophagy inducers, Bioorganic & Medicinal Chemistry Letters 2011, 21, 234-239.
  36. Han, Shuai; Pan, Heling; Zhang, Jianhua; Tan, Li; Ma, Dawei*; Yuan, Junying; Wu, Jia-Rui Identification of a small molecule activator of novel PKCs for promoting glucose-dependent insulin secretion, Cell Research 2011, 21, 588-599.
  37. Li, Wenhua; Yu, Shouyun; Jin, Mingzhi; Xia, Hongguang; Ma, Dawei* Total synthesis and cytotoxicity of bisebromoamide and its analogues, Tetrahedron Letters 2011, 52, 2124-2127.
  38. Liu, Junli; Xia, Hongguang; Kim, Minsu; Xu, Lihua; Li, Ying; Zhang, Lihong; Cai, Yu; Norberg, Helin Vakifahmetoglu; Zhang, Tao; Furuya, Tsuyoshi; Jin, Minzhi; Zhu, Zhimin; Wang, Huanchen; Yu, Jia; Li, Yanxia; Hao, Yan; Choi, Augustine; Ke, Hengming; Ma, Dawei*; Yuan, Junying Beclin1 Controls the Levels of p53 by Regulating the Deubiquitination Activity of USP10 and USP13, Cell (Cambridge, MA, United States) 2011, 147, 223-234.
  39. Ma, Dawei*; Jiang, Yongwen Cu(I)/amino acid catalyzed coupling reactions of aryl halides and nucleophiles: applications in large-scale production, Chimia 2011, 65, 914-918.
  40. Ma, Dawei*; Lu, Xu; Shi, Liu; Zhang, Hui; Jiang, Yongwen; Liu, Xiangqian Domino condensation/S-arylation/heterocyclization reactions: copper-catalyzed three-component synthesis of 2-N-substituted benzothiazoles, Angewandte Chemie, International Edition 2011, 50, 1118-1121.
  41. Shi, Liu; Liu, Xiangqian; Zhang, Hui; Jiang, Yongwen; Ma, Dawei* Synthesis of 2-thio-substituted benzothiazoles via a domino condensation/S-arylation/heterocyclization process, Journal of Organic Chemistry 2011, 76, 4200-4204.
  42. Sun, Xuefeng; Ma, Dawei* Organocatalytic Approach for the Syntheses of Corynantheidol, Dihydrocorynantheol, Protoemetinol, Protoemetine, and Mitragynine, Chemistry--An Asian Journal, 2011, 6, 2158-2165.
  43. Wang, You; Zhu, Shaolin; Ma, Dawei* Organocatalytic Approach to Polysubstituted Piperidines and Tetrahydropyrans, Organic Letters 2011, 13, 1602-1605.
  44. Yu, Shouyun; Zhu, Shaolin; Pan, Xianhua; Yang, Jiade; Ma, Dawei* Reinvestigation on total synthesis of kaitocephalin and its isomers, Tetrahedron 2011, 67, 1673-1680.
  45. Zuo, Zhiwei; Ma, Dawei* Enantioselective Total Syntheses of Communesins A and B, Angewandte Chemie, International Edition 2011, 50, 12008-12011.
  46. Zuo, Zhiwei; Ma, Dawei* Synthetic studies toward communesins, Israel Journal of Chemistry 2011, 51, 434-441.
  47. Zi Weiwei, Yu Shouyun and Ma Dawei*, A convergent route to galbulimima alkaloid (-)-GB 13 and (+)-GB 16, Angewandte Chemie, International Edition 2010, 49, 5887.
  48. Chang M., Kanwar N., Feng E., Siu A., Liu X., Ma D., Jongstra J., PIM kinase inhibitors downregulate STAT3Tyr705 phosphorylation. Mol. Cancer Ther. 2010, 9,2478.
  49. Ben, Li; Jones, Eric Dale; Zhou, Enkun; Li, Chen; Baylis, Dean Cameron; Yu, Shanghai; Wang, Miao; He, Xing; Coates, Jonathan Alan Victor; Rhodes, David Ian; Pei, Gang; Deadman, John Joseph; Xie, Xin; Ma, Dawei Studies on the structure-activity relationship of 1,3,3,4-tetra-substituted pyrrolidine embodied CCR5 receptor antagonists. Part 1: Tuning the N-substituents, Bioorganic & Medicinal Chemistry Letters 2010, 20, 4012-4014.
  50. Hao, Chao; Zhang, Yihua; Jiang, Yongwen; Ma, Dawei* CuBr/N,N-dimethylglycine-catalyzed coupling reaction of 2-chlorotrifluoroacetanilides with phenols at mild conditions, Chinese Journal of Chemistry 2010, 28, 1645-1650.
  51. Li, Ben; Jones, Eric Dale; Zhou, Enkun; Chen, Li; Baylis, Dean Cameron; Yu, Shanghai; Wang, Miao; He, Xing; Coates, Jonathan Alan Victor; Rhodes, David Ian; Pei, Gang; Deadman, John Joseph; Xie, Xin; Ma, Dawei* Studies on the structure-activity relationship of 1,3,3,4-tetra-substituted pyrrolidine embodied CCR5 receptor antagonists. Part 2: Discovery of highly potent anti-HIV agents, Bioorganic & Medicinal Chemistry Letters 2010, 20, 5334-5336.
  52. Li, Wenhua; Schlecker, Andreas; Ma, Dawei* Total synthesis of antimicrobial and antitumor cyclic depsipeptides, Chemical Communications (Cambridge, United Kingdom) 2010, 46, 5403-5420.
  53. Lu, Xu; Shi, Liu; Zhang, Hui; Jiang, Yongwen; Ma, Dawei* Assembly of N-substituted pyrrolo[2,1-c][1,4]benzodiazepine-5,11-diones via copper catalyzed aryl amination, Tetrahedron 2010, 66, 5714-5718.
  54. Ma, Anqi; Ma, Dawei* Enantioselective Synthesis of Polysubstituted Cyclopentanones by Organocatalytic Double Michael Addition Reactions, Organic Letters 2010, 12, 3634-3637.
  55. Ma, Dawei*; Geng, Qian; Zhang, Hui; Jiang, Yongwen Assembly of Substituted Phenothiazines by a Sequentially Controlled CuI/L-Proline-Catalyzed Cascade C-S and C-N Bond Formation, Angewandte Chemie, International Edition 2010, 49, 1291-1294.
  56. Maurer, Stefan; Liu, Wei; Zhang, Xiaojing; Jiang, Yongwen; Ma, Dawei* An efficient synthesis of phenol via CuI/8-hydroxyquinoline-catalyzed hydroxylation of aryl halides and potassium hydroxide, Synlett 2010, 976-978.
  57. Wang, You; Xu, Lanting; Ma, Dawei* CuI/L-Proline-Catalyzed Coupling of Substituted 3-Iodoprop-2-en-1-ols with 1-Alkynes and Subsequent Cyclization: A Convenient Approach for Synthesizing Polysubstituted Furans, Chemistry--An Asian Journal 2010, 5, 74-76.
  58. Xia, Hong-guang; Zhang, Lihong; Chen, Gang; Zhang, Tao; Liu, Junli; Jin, Mingzhi; Ma, Xiuquan; Ma, Dawei*; Yuan, Junying Control of basal autophagy by calpain1 mediated cleavage of ATG5, Autophagy 2010, 6, 61-66.
  59. Xu, Danhua; Zhang, Yihua; Ma, Dawei* Organocatalytic approach to 3,5,6-trisubstituted and 4,6-disubstituted tetrahydropyran-2-ones, Tetrahedron Letters 2010, 51, 3827-3829.
  60. Xu, Lanting; Jiang, Yongwen; Ma, Dawei* Synthesis of tetrahydropyrrolo[1,2-a]quinoxalines and tetrahydropyrido[1,2-a]quinoxalines via a one-pot CuI-catalyzed aryl amination-hydrolysis-condensation process, Synlett, 2010, 2285-2288.
  61. Zhou, Qianghui; Chen, Xiaofei; Ma, Dawei Asymmetric, Protecting-Group-Free Total Synthesis of (-)-Englerin A, Angewandte Chemie, International Edition 2010, 49, 3513-3516.
  62. Zhu, Shaolin; Yu, Shouyun; Wang, You; Ma, Dawei* Organocatalytic Michael addition of aldehydes to protected 2-amino-1-nitroethenes: the practical syntheses of oseltamivir (Tamiflu) and substituted 3-aminopyrrolidines, Angewandte Chemie, International Edition 2010, 49, 4656-4660.
  63. Zi, Weiwei; Yu, Shouyun; Ma, Dawei* A Convergent Route to the Galbulimima Alkaloids (-)-GB 13 and (+)-GB 16, Angewandte Chemie, International Edition 2010, 49, 5887-5890.
  64. Zi, Weiwei; Yu, Shouyun; Ma, Dawei* Synthetic Studies toward Galbulimima Alkaloid (-)-GB 13 and (+)-GB 16 and (-)-Himgaline, Chemistry, an Asian journal 2010,6,573.
  65. Zuo, Zhiwei; Xie, Weiqing; Ma, Dawei* Total Synthesis and Absolute Stereochemical Assignment of (-)-Communesin F, Journal of the American Chemical Society 2010, 132, 13226-13228.
发表时间:2015-03-01 阅读次数:1679次

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